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Lefamulin acetate

Glpbio
Catalog No:GC39163-10mM (in 1mL DMSO) CAS No.:1350636-82-6 MDLNo: Brand:Glpbio purity: 特性: Purpose:Lefamulin acetate (BC-3781 acetate) 是一種口服活性抗生素,用于 community-acquired bacterial pneumonia (CABP) 治療。Lefamulin acetate (BC-3781 acetate) 是第一種用于人體細(xì)菌感染的全身治療的半合成截短側(cè)耳素。Lefamulin acetate (BC-3781 acetate) 通過與 50S 細(xì)菌核糖體的肽基轉(zhuǎn)移酶 peptidyl transferase 中心結(jié)合來抑制蛋白質(zhì)合成,從而阻止了轉(zhuǎn)移RNA與肽轉(zhuǎn)移的結(jié)合。DMSO: ≥ 100 mg/mL (176.12 mM); H2O: < 0.1 mg/mL (insoluble)
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